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現(xiàn)貨moradec AH-207-DX說明書

 更新時(shí)間:2022-12-28 點(diǎn)擊量:825


現(xiàn)貨moradec AH-207-DX說明書


Fab-αHFc-CL-DX8951

Fab抗人IgG Fc-DX9851抗體

目錄號:AH-207-DX

Fab-αHFc-CL-DX8951是抗人IgG Fc特異性抗體的Fab片段,與甲磺酸艾替康(DX8951)結(jié)合,具有可裂解的接頭。抗體部分是對人IgG的Fc區(qū)特異的多克隆抗體Fab片段。甲磺酸埃克替康(DX8951)是一種拓?fù)洚悩?gòu)酶I抑制劑。連接DX8951和抗體的可裂解接頭(GGFG)在細(xì)胞外液中是穩(wěn)定的,但一旦綴合物通過內(nèi)吞作用進(jìn)入細(xì)胞,就會(huì)在內(nèi)體中被裂解。Fab 2°ADC的單價(jià)性質(zhì)在某些應(yīng)用中可能比全長IgG 2°ADC具有一些優(yōu)勢。



Fab-αHFc-CL-DX8951


Fab Anti-Human IgG Fc-DX9851 Antibody with Cleavable Linker

Catalog Number: AH-207-DX

Fab-αHFc-CL-DX8951 is a Fab fragment of anti-human IgG Fc specific antibody conjugated to exatecan mesylate (DX8951) with a cleavable linker. The antibody portion is a polyclonal antibody Fab fragment specific to the Fc region of human IgGs. Exatecan mesylate (DX8951) is a topoisomerase I inhibitor. The cleavable linker (GGFG) connecting DX8951 to the antibody is stable in extracellular fluid, but is cleaved by in endosome once the conjugate has entered a cell via endocytosis.The mono-valence nature of Fab 2°ADC may have some advantage in certain applications than the full length IgG 2°ADC.